PDB: 6LIL
Title: Crystal structure of human PDK2 complexed with an allosteric inhibitor compound 8c
PDB: 6LIN
Title: Crystal structure of human PDK2 complexed with GM10030
PDB: 6LIO
Title: Crystal structure of human PDK2 complexed with GM67520
Publication
Structural basis for the inhibition of PDK2 by novel ATP- and lipoyl-binding site targeting compounds
Author : Jihoon Kang, Haushabhau S. Pagire, Donguk Kang, Yo Han Song, In Kyu Lee, Kang Taek Lee, Chin-Ju Park, Jin Hee Ahn, and Jungwook Kim
Biochem Biophys Res Commun. 2020 Jun 30;527(3):778-784. doi: 10.1016/j.bbrc.2020.04.102
